BRL 44408 maleate | Tocris Bioscience 1133 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

BRL 44408 maleate

catalog :

1133

quantity :

10 mg (also 50 mg)

price :

173 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Rennekamp A, Huang X, Wang Y, Patel S, Lorello P, Cade L, et al. ?1 receptor ligands control a switch between passive and active threat responses. Nat Chem Biol. 2016;12:552-8 pubmed publisher
Backman L, Andersson G, Fong G, Alfredson H, Scott A, Danielson P. Alpha-2 adrenergic stimulation triggers Achilles tenocyte hypercellularity: Comparison between two model systems. Scand J Med Sci Sports. 2013;23:687-96 pubmed publisher

product information

brand :

Tocris

master code :

1133

SKU :

1133/10

product name :

BRL 44408 maleate

description :

Selective 2A antagonist

target :

Adrenergic alpha-2 Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

331.37

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Selective 2A-adrenoceptor antagonist (Ki = 1.7 nM and 144.5 nM at 2A and 2B-adrenergic receptors respectively). Increases hippocampal noradrenalin release following systemic administration. Also available as part of the 2 -Adrenoceptor Tocriset .

catalog number base :

1133

product keywords :

Selective alpha2A-adrenoceptor a2a-adrenoceptor a2a-Adrenergic a2a-adrenergic antagonists Receptors BRL44408 maleate GlaxoSmithKline GSK Adrenergic Alpha-2 Receptors 1133,

extended description :

Selective 2A antagonist

chemical name text :

2-[(4,5-Dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole maleate

formula :

C 13 H 17 N 3 .C 4 H 4 O 4

formula text :

C13H17N3.C4H4O4

cas num :

681806-46-2

2020 USD :

166

2021 USD :

173 USD

storage :

Desiccate at -20°C

more info or order :

Tocris Bioscience product webpage