1133/10 | Tocris Bioscience 1133/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

1133/10

catalog :

1133/10

quantity :

10 mg (also 50 mg)

price :

195 USD

more info or order :

Tocris Bioscience product webpage

citations: 3

Reference
Rennekamp A, Huang X, Wang Y, Patel S, Lorello P, Cade L, et al. ?1 receptor ligands control a switch between passive and active threat responses. Nat Chem Biol. 2016;12:552-8 pubmed publisher
Fox J, Sakamuru S, Huang R, Teneva N, Simmons S, Xia M, et al. High-throughput genotoxicity assay identifies antioxidants as inducers of DNA damage response and cell death. Proc Natl Acad Sci U S A. 2012;109:5423-8 pubmed publisher
Backman L, Andersson G, Fong G, Alfredson H, Scott A, Danielson P. Alpha-2 adrenergic stimulation triggers Achilles tenocyte hypercellularity: Comparison between two model systems. Scand J Med Sci Sports. 2013;23:687-96 pubmed publisher

product information

master code :

1133

SKU :

1133/10

product name :

BRL 44408 maleate

unit size :

10 mg (also 50 mg)

description :

Selective 2A antagonist

target :

Adrenergic alpha-2 Receptor Antagonists

category :

Small Molecules

purity :

98%

observed molecular weight :

331.37

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

BRL 44408 maleate is a selective 2A-adrenoceptor antagonist (Ki = 1.7 nM and 144.5 nM at 2A and 2B-adrenergic receptors respectively). Increases hippocampal noradrenalin release following systemic administration.

top caption :

Selective 2A antagonist

extended description :

Selective 2A antagonist

chemical name text :

2-[(4,5-Dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole maleate

formula :

C13H17N3.C4H4O4

formula text :

C13H17N3.C4H4O4

cas num :

681806-46-2

USD :

195 USD

product details :

Selective 2A antagonist

storage :

Desiccate at -20░C

more info or order :

Tocris Bioscience product webpage