1122/10 | Tocris Bioscience 1122/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

1122/10

catalog :

1122/10

quantity :

10 mg (also 50 mg)

price :

86 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Pediani J, Ward R, Godin A, Marsango S, Milligan G. Dynamic Regulation of Quaternary Organization of the M1 Muscarinic Receptor by Subtype-selective Antagonist Drugs. J Biol Chem. 2016;291:13132-46 pubmed publisher
Fox J, Sakamuru S, Huang R, Teneva N, Simmons S, Xia M, et al. High-throughput genotoxicity assay identifies antioxidants as inducers of DNA damage response and cell death. Proc Natl Acad Sci U S A. 2012;109:5423-8 pubmed publisher

image

image 1 :

Cat.No. 1122 - Telenzepine dihydrochloride C19H22N4O2S.2HCl CAS No. 147416-96-4

product information

master code :

1122

SKU :

1122/10

product name :

Telenzepine dihydrochloride

unit size :

10 mg (also 50 mg)

description :

Potent, selective M1 antagonist

target :

mAChR M1 Antagonists

category :

Small Molecules

purity :

98%

observed molecular weight :

443.39

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Telenzepine dihydrochloride is a selective high affinity muscarinic M1 receptor antagonist (Ki = 0.94 nM). Inhibits gastric acid secretion.

top caption :

Potent, selective M1 antagonist

extended description :

Potent, selective M1 antagonist

chemical name text :

4,9-Dihydro-3-methyl-4-[(4-methyl-1-piperazinyl)acetyl]-10H-thieno[3,4-b][1,5]benzodiazepin-10-one dihydrochloride

formula :

C19H22N4O2S.2HCl

formula text :

C19H22N4O2S.2HCl

cas num :

147416-96-4

USD :

86 USD

product details :

Potent, selective M1 antagonist

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage