LY 225910 | Tocris Bioscience 1018 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

LY 225910

catalog :

1018

quantity :

10 mg (also 50 mg)

price :

115 USD

more info or order :

Tocris Bioscience product webpage

citations: 3

Reference
Seillier A, Martinez A, Giuffrida A. Phencyclidine-induced social withdrawal results from deficient stimulation of cannabinoid CB? receptors: implications for schizophrenia. Neuropsychopharmacology. 2013;38:1816-24 pubmed publisher
Karson M, Whittington K, Alger B. Cholecystokinin inhibits endocannabinoid-sensitive hippocampal IPSPs and stimulates others. Neuropharmacology. 2008;54:117-28 pubmed
Gallopin T, Geoffroy H, Rossier J, Lambolez B. Cortical sources of CRF, NKB, and CCK and their effects on pyramidal cells in the neocortex. Cereb Cortex. 2006;16:1440-52 pubmed

product information

brand :

Tocris

master code :

1018

SKU :

1018/10

product name :

LY 225910

description :

Potent CCK2 antagonist

target :

CCK2 Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

observed molecular weight :

502.41

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent CCK2 receptor antagonist (IC50 = 9.3 nM for inhibition of 125I-labeled CCK-8 sulfate binding at mouse brain membranes).

catalog number base :

1018

product keywords :

Potent CCK2 antagonists Cholecystokinin2 Receptors LY225910 CCK2 Receptor 1018,

extended description :

Potent CCK2 antagonist

chemical name text :

2-[2-(5-Bromo-1H-indol-3-yl)ethyl]-3-[3-(1-methylethoxy)phenyl]-4-(3H)-quinazoline

formula :

C 27 H 24 BrN 3 O 2

formula text :

C27H24BrN3O2

cas num :

133040-77-4

2020 USD :

112

2021 USD :

115 USD

storage :

Desiccate at -20°C

more info or order :

Tocris Bioscience product webpage