Cyanopindolol hemifumarate | Tocris Bioscience 0993 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Cyanopindolol hemifumarate

catalog :

0993

quantity :

10 mg (also 50 mg)

price :

169 USD

more info or order :

Tocris Bioscience product webpage

citations: 4

Reference
Gautam J, Banskota S, Regmi S, Ahn S, Jeon Y, Jeong H, et al. Tryptophan hydroxylase 1 and 5-HT7 receptor preferentially expressed in triple-negative breast cancer promote cancer progression through autocrine serotonin signaling. Mol Cancer. 2016;15:75 pubmed
Kaya A, Ugur O, Oner S, Bastepe M, Onaran H. Coupling of beta2-adrenoceptors to XLalphas and Galphas: a new insight into ligand-induced G protein activation. J Pharmacol Exp Ther. 2009;329:350-9 pubmed publisher
Brahmadevara N, Shaw A, Macdonald A. ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta. Br J Pharmacol. 2004;142:781-7 pubmed
Geerts I, Matthys K, Herman A, Bult H. Involvement of 5-HT1B receptors in collar-induced hypersensitivity to 5-hydroxytryptamine of the rabbit carotid artery. Br J Pharmacol. 1999;127:1327-36 pubmed

product information

brand :

Tocris

master code :

0993

SKU :

0993/10

product name :

Cyanopindolol hemifumarate

description :

5-HT1A and 5-HT1B antagonist; also -adrenergic antagonist

target :

5-HT1A Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

345.4

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

5-HT1A/1B antagonist with roughly equal affinity at each receptor; also a -adrenoceptor antagonist.

catalog number base :

993

product keywords :

5-HT1A/1B antagonists -adrenergic beta-adrenergic -adrenoceptor beta-adrenoceptor b-adrenergic b-adrenoceptor Serotonin 5-HT1A Receptors 5-HT1A Receptors 5-HT1B Receptors Non-selective Adrenergic Beta Receptors 0993,

extended description :

5-HT1A and 5-HT1B antagonist; also -adrenergic antagonist

chemical name text :

4-[3-[tert-Butylamino]-2-hydroxypropoxy]-1H-indole-2-carbonitrile hemifumarate

formula :

C 16 H 21 N 3 O 2 . C 4 H 4 O 4

formula text :

C16H21N3O2.?C4H4O4

cas num :

69906-86-1

2020 USD :

164

2021 USD :

169 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage