Remoxipride hydrochloride | Tocris Bioscience 0916 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Remoxipride hydrochloride

catalog :

0916

quantity :

10 mg (also 50 mg)

price :

159 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Andre V, Cepeda C, Fisher Y, Huynh M, Bardakjian N, Singh S, et al. Differential electrophysiological changes in striatal output neurons in Huntington's disease. J Neurosci. 2011;31:1170-82 pubmed publisher

product information

brand :

Tocris

master code :

0916

SKU :

0916/10

product name :

Remoxipride hydrochloride

description :

Selective D2-like antagonist

target :

Non-selective Dopamine Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

observed molecular weight :

407.73

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Dopamine D2 receptor antagonist showing selectivity over D3 and D4 receptors (Ki values are ~ 300, ~ 1600, and ~ 2800 nM for D2, D3 and D4 receptors respectively). Exhibits antipsychotic activity in vivo with no extrapyramidal side effects. 50-fold more potent than sulpiride in antagonising the effects of apomorphine in the rat.

catalog number base :

916

product keywords :

selective D2-like antagonists dopamine non-selective receptor antagonist dopaminergic d2 Non-selective Dopamine 0916,

extended description :

Selective D2-like antagonist

chemical name text :

(S)-(-)-3-Bromo-N-[(1-ethyl-2-pyrrolidinylmethyl]2,6-dimethoxybenzamide hydrochloride

formula :

C 16 H 23 BrN 2 O 3 .HCl

formula text :

C16H23BrN2O3.HCl

cas num :

73220-03-8

2020 USD :

154

2021 USD :

159 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage