L-732,138 | Tocris Bioscience 0868 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

L-732,138

catalog :

0868

quantity :

10 mg (also 50 mg)

price :

95 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Wan F, Bai Y, Kou Z, Zhang T, Li H, Wang Y, et al. Endomorphin-2 Inhibition of Substance P Signaling within Lamina I of the Spinal Cord Is Impaired in Diabetic Neuropathic Pain Rats. Front Mol Neurosci. 2016;9:167 pubmed publisher
Li X, Ma G, Ma Q, Li W, Liu J, Han L, et al. Neurotransmitter substance P mediates pancreatic cancer perineural invasion via NK-1R in cancer cells. Mol Cancer Res. 2013;11:294-302 pubmed publisher

product information

brand :

Tocris

master code :

0868

SKU :

0868/10

product name :

L-732,138

description :

Potent and selective NK1 antagonist

target :

NK1 Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

472.39

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and highly selective competitive tachykinin NK1 receptor antagonist (IC50 = 2.3 nM).

catalog number base :

868

product keywords :

Potent selective NK1 antagonists Tachykinin Receptors Neurokinin L732138 merck NK1 Receptor 0868, Neurokinin NK1

extended description :

Potent and selective NK1 antagonist

chemical name text :

N-Acetyl-L-tryptophan 3,5-bis(trifluoromethyl)benzyl ester

formula :

C 22 H 18 F 6 N 2 O 3

formula text :

C22H18F6N2O3

cas num :

148451-96-1

2020 USD :

2021 USD :

95 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage