Rilmenidine hemifumarate | Tocris Bioscience 0790 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Rilmenidine hemifumarate

catalog :

0790

quantity :

25 mg

price :

324 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Sánchez Blázquez P, Boronat M, Olmos G, García Sevilla J, Garzon J. Activation of I(2)-imidazoline receptors enhances supraspinal morphine analgesia in mice: a model to detect agonist and antagonist activities at these receptors. Br J Pharmacol. 2000;130:146-52 pubmed

product information

brand :

Tocris

master code :

0790

SKU :

0790/25

product name :

Rilmenidine hemifumarate

description :

2 agonist. Also I1 ligand

target :

Adrenergic alpha-2 Receptor Agonists

category :

Small Molecules

unit size :

25 mg

purity :

99%

observed molecular weight :

238.29

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

I1-imidazoline binding site selective ligand and 2-adrenoceptor agonist. Possesses greater I1 vs 2 selectivity than the prototypical compound, clonidine. Also thought to enhance autophagy; shown to increase LC3-II levels in PC12 cells.

catalog number base :

790

product keywords :

2-adrenoceptor alpha2-adrenoceptor a2-adrenoceptor 2-Adrenergic alpha2-Adrenergic a2-adrenergic agonists I1 ligand Receptors Imidazoline Adrenergic Alpha-2 Receptors I1 Receptors Autophagy 0790,

extended description :

2 agonist. Also I1 ligand

chemical name text :

2-[N-(Dicyclopropylmethyl)amino]oxazoline hemifumarate

formula :

C 10 H 16 N 2 O. C 4 H 4 O 4

formula text :

C10H16N2O.?C4H4O4

cas num :

207572-68-7

2020 USD :

308

2021 USD :

324 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage