0790/5 | Tocris Bioscience 0790/5 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

0790/5

catalog :

0790/5

quantity :

5 mg (also 25 mg)

price :

111 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Fox J, Sakamuru S, Huang R, Teneva N, Simmons S, Xia M, et al. High-throughput genotoxicity assay identifies antioxidants as inducers of DNA damage response and cell death. Proc Natl Acad Sci U S A. 2012;109:5423-8 pubmed publisher
Sánchez Blázquez P, Boronat M, Olmos G, García Sevilla J, Garzon J. Activation of I(2)-imidazoline receptors enhances supraspinal morphine analgesia in mice: a model to detect agonist and antagonist activities at these receptors. Br J Pharmacol. 2000;130:146-52 pubmed

product information

master code :

790

SKU :

0790/5

product name :

Rilmenidine hemifumarate

unit size :

5 mg (also 25 mg)

description :

I1 ligand. Also 2 agonist

target :

Adrenergic alpha-2 Receptor Agonists

category :

Small Molecules

purity :

98%

observed molecular weight :

238.29

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Rilmenidine hemifumarate is an I1-imidazoline binding site selective ligand and 2-adrenoceptor agonist. Possesses greater I1 vs 2 selectivity than the prototypical compound, clonidine. Also thought to enhance autophagy; shown to increase LC3-II levels in PC12 cells.

top caption :

I1 ligand. Also 2 agonist

extended description :

I1 ligand. Also 2 agonist

chemical name text :

2-[N-(Dicyclopropylmethyl)amino]oxazoline hemifumarate

formula :

C10H16N2O. C4H4O4

formula text :

C10H16N2O.?C4H4O4

cas num :

207572-68-7

USD :

111 USD

product details :

I1 ligand. Also 2 agonist

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage