Amthamine dihydrobromide | Tocris Bioscience 0668 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Amthamine dihydrobromide

catalog :

0668

quantity :

10 mg (also 50 mg)

price :

161 USD

more info or order :

Tocris Bioscience product webpage

citations: 4

Reference
Saligrama N, Case L, Krementsov D, Teuscher C. Histamine H₂ receptor signaling × environment interactions determine susceptibility to experimental allergic encephalomyelitis. FASEB J. 2014;28:1898-909 pubmed publisher
Chigaev A, Smagley Y, Zhang Y, Waller A, Haynes M, Amit O, et al. Real-time analysis of the inside-out regulation of lymphocyte function-associated antigen-1 revealed similarities to and differences from very late antigen-4. J Biol Chem. 2011;286:20375-86 pubmed publisher
Copsel S, Garcia C, Diez F, Vermeulem M, Baldi A, Bianciotti L, et al. Multidrug resistance protein 4 (MRP4/ABCC4) regulates cAMP cellular levels and controls human leukemia cell proliferation and differentiation. J Biol Chem. 2011;286:6979-88 pubmed publisher
Flamand N, Plante H, Picard S, Laviolette M, Borgeat P. Histamine-induced inhibition of leukotriene biosynthesis in human neutrophils: involvement of the H2 receptor and cAMP. Br J Pharmacol. 2004;141:552-61 pubmed

product information

brand :

Tocris

master code :

0668

SKU :

0668/10

product name :

Amthamine dihydrobromide

description :

Highly selective standard H2 agonist

target :

Histamine H2 Receptor Agonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

319.06

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Highly selective H2 agonist, slightly more potent than histamine itself. Only a weak antagonist at H3 and has no activity at H1 receptors. Induces vasodilation of cerebral arteries and decreases myogenic tone in vitro .

catalog number base :

668

product keywords :

selective H2 agonists Receptors Histamine histaminergic Histamine H2 Receptors 0668,

extended description :

Highly selective standard H2 agonist

chemical name text :

2-Amino-5-(2-aminoethyl)-4-methylthiazole dihydrobromide

formula :

C 6 H 11 N 3 S.2HBr

formula text :

C6H11N3S.2HBr

cas num :

142457-00-9

2020 USD :

154

2021 USD :

161 USD

storage :

Desiccate at -20°C

more info or order :

Tocris Bioscience product webpage