4F 4PP oxalate | Tocris Bioscience 0523 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

4F 4PP oxalate

catalog :

0523

quantity :

10 mg (also 50 mg)

price :

158 USD

more info or order :

Tocris Bioscience product webpage

citations: 3

Reference
Lee S, Cho P, Tonello R, Lee H, Jang J, Park G, et al. Peripheral serotonin receptor 2B and transient receptor potential channel 4 mediate pruritus to serotonergic antidepressants in mice. J Allergy Clin Immunol. 2018;: pubmed publisher
Rodríguez Muñoz M, Sánchez Blázquez P, Garzón J. Fenfluramine diminishes NMDA receptor-mediated seizures via its mixed activity at serotonin 5HT2A and type 1 sigma receptors. Oncotarget. 2018;9:23373-23389 pubmed publisher
Gerhold K, Drdla Schutting R, Honsek S, Forsthuber L, SandkÃ¼hler J. Pronociceptive and Antinociceptive Effects of Buprenorphine in the Spinal Cord Dorsal Horn Cover a Dose Range of Four Orders of Magnitude. J Neurosci. 2015;35:9580-94 pubmed publisher

product information

brand :

Tocris

master code :

0523

SKU :

0523/10

product name :

4F 4PP oxalate

description :

Selective 5-HT2A antagonist

target :

5-HT2A Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

429.49

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

A selective 5-HT2A antagonist with almost as high affinity (Ki = 5.3 nM) as ketanserin but with a much lower affinity for 5-HT2C sites (Ki = 620 nM).

catalog number base :

523

product keywords :

Selective 5-HT2A antagonists Serotonin Receptors 5-HT2 4F4PP oxalate 5-HT2A Receptors 0523,

extended description :

Selective 5-HT2A antagonist

chemical name text :

4-(4-Fluorobenzoyl)-1-(4-phenylbutyl)piperidine oxalate

formula :

C 22 H 26 FNO.C 2 H 2 O 4

formula text :

C22H26FNO.C2H2O4

cas num :

144734-36-1

2020 USD :

154

2021 USD :

158 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage