0307/10 | Tocris Bioscience 0307/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

0307/10

catalog :

0307/10

quantity :

10 mg (also 50 mg)

price :

174 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Pollok S, Reiner A. Subunit-selective iGluR antagonists can potentiate heteromeric receptor responses by blocking desensitization. Proc Natl Acad Sci U S A. 2020;117:25851-25858 pubmed publisher
Pansiot J, Loron G, Olivier P, Fontaine R, Charriaut Marlangue C, Mercier J, et al. Neuroprotective effect of inhaled nitric oxide on excitotoxic-induced brain damage in neonatal rat. PLoS ONE. 2010;5:e10916 pubmed publisher

product information

master code :

307

SKU :

0307/10

product name :

(S)-(-)-5-Iodowillardiine

unit size :

10 mg (also 50 mg)

description :

Highly potent and subtype-selective kainate agonist

target :

Kainate Receptor Agonists

category :

Small Molecules

purity :

98%

observed molecular weight :

325.06

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Demonstrates high affinity for the kainate receptor subtype hGluK1 (formerly hGluR5) (Ki = 0.24 nM) and 600-4000-fold selectivity over both the AMPA receptor subtypes and the homomeric kainate receptor hGluK2 (formerly hGluR6). . Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions .

top caption :

Highly potent and subtype-selective kainate agonist

extended description :

Highly potent and subtype-selective kainate agonist

formula :

C7H8IN3O4

formula text :

C7H8IN3O4

cas num :

140187-25-3

USD :

174 USD

product details :

Highly potent and subtype-selective kainate agonist

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage