Src I1 | Enzo Life Sciences BML-EI398-0025 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Enzo Life Sciences

other brands :

Stressgen, BioMol, Alexis Corporation, Assay Designs, Alexis

product type :

chemical

product name :

Src I1

catalog :

BML-EI398-0025

quantity :

25 mg

citations: 2

Reference
Bain J, Plater L, Elliott M, Shpiro N, Hastie C, McLauchlan H, et al. The selectivity of protein kinase inhibitors: a further update. Biochem J. 2007;408:297-315 pubmed
Tian G, Cory M, Smith A, Knight W. Structural determinants for potent, selective dual site inhibition of human pp60c-src by 4-anilinoquinazolines. Biochemistry. 2001;40:7084-91 pubmed

product information

Product ID :

BML-EI398

Catalog Number :

BML-EI398-0025

Product Name :

Src I1

Product Type :

Biochemical

Size :

25 mg

list of Pubmed id :

17850214, 11401553

Product Description :

Potent, dual site (ATP domain and substrate-binding domain) Src and Lck kinase inhibitor (IC50=44 and 88nM respectively). VEGFR2 IC50=0.32μM; c-fms IC50=30μM.

ALTnames :

6,7-Dimethoxy-N-(4-phenoxyphenyl)-4-quinazolinamine

Purity :

≥98% (HPLC)

Storage :

Ambient